Title : Phase 1 summary of plasma concentration-QTc analysis for idasanutlin, an MDM2 antagonist, in patients with advanced solid tumors and AML.

Pub. Date : 2018 Mar

PMID : 29392451






2 Functional Relationships(s)
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1 PURPOSE: Idasanutlin, a selective small-molecule MDM2 antagonist in phase 3 testing for refractory/relapsed AML, is a non-genotoxic oral p53 activator. RG7388 MDM2 proto-oncogene Homo sapiens
2 Phase 1 summary of plasma concentration-QTc analysis for idasanutlin, an MDM2 antagonist, in patients with advanced solid tumors and AML. RG7388 MDM2 proto-oncogene Homo sapiens