Title : Modulation of CYP3A enzyme activity by diosmin and its consequence on carbamazepine pharmacokinetics in rats.

Pub. Date : 2018 Feb

PMID : 29134244






2 Functional Relationships(s)
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1 Diosmin-mediated altered CYP3A enzyme activity in human and rat liver microsomes was examined using CYP3A dependent erythromycin N-demethylase assay. Diosmin cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 The CYP3A enzyme activity in human and rat liver microsomes was significantly (p < 0.05) decreased by diosmin when compared to control. Diosmin cytochrome P450 family 3 subfamily A member 4 Homo sapiens