Title : The potential of natural products for targeting PPARα.

Pub. Date : 2017 Jul

PMID : 28752027






1 Functional Relationships(s)
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1 PPARs constitute a recognized druggable target and indeed several classes of drugs used in the treatment of metabolic disease symptoms, such as dyslipidemia (fibrates, e.g. fenofibrate and gemfibrozil) and diabetes (thiazolidinediones, e.g. rosiglitazone and pioglitazone) are ligands for the various PPAR isoforms. Gemfibrozil peroxisome proliferator activated receptor alpha Homo sapiens