Title : Discovery and Characterization of 1H-Pyrazol-5-yl-2-phenylacetamides as Novel, Non-Urea-Containing GIRK1/2 Potassium Channel Activators.

Pub. Date : 2017 Sep 20

PMID : 28697302






2 Functional Relationships(s)
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1 Discovery and Characterization of 1H-Pyrazol-5-yl-2-phenylacetamides as Novel, Non-Urea-Containing GIRK1/2 Potassium Channel Activators. Urea potassium inwardly rectifying channel subfamily J member 3 Homo sapiens
2 Previously reported urea containing molecules as GIRK1/2 preferring activators have had significant pharmacokinetic (PK) liabilities. Urea potassium inwardly rectifying channel subfamily J member 3 Homo sapiens