Title : Development of Selective Clk1 and -4 Inhibitors for Cellular Depletion of Cancer-Relevant Proteins.

Pub. Date : 2017 Jul 13

PMID : 28561591






1 Functional Relationships(s)
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1 On the basis of a Weinreb amide hit compound, we designed and synthesized a diverse set of methoxybenzothiophene-2-carboxamides, of which the N-benzylated derivative showed enhanced Clk1 inhibitory activity. weinreb amide CDC like kinase 1 Homo sapiens