Title : Identification of a novel 5-amino-3-(5-cyclopropylisoxazol-3-yl)-1-isopropyl-1H-pyrazole-4-carboxamide as a specific RET kinase inhibitor.

Pub. Date : 2017 Jan 5

PMID : 27814560






1 Functional Relationships(s)
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1 In a recent effort we identified a novel and specific RET inhibitor of 5-aminopyrazole-4-carboxamide scaffold, which was designed to enhance the metabolic stability of the pyrazolopyrimidine scaffold. 3-Amino-1H-pyrazole-4-carboxamide ret proto-oncogene Homo sapiens