Pub. Date : 2016 Dec
PMID : 27751847
8 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
1 | Osimertinib for pretreated EGFR Thr790Met-positive advanced non-small-cell lung cancer (AURA2): a multicentre, open-label, single-arm, phase 2 study. | osimertinib | epidermal growth factor receptor | Homo sapiens |
2 | BACKGROUND: Osimertinib (AZD9291) is an oral, potent, irreversible EGFR tyrosine-kinase inhibitor selective for EGFR tyrosine-kinase inhibitor sensitising mutations, and the EGFR Thr790Met resistance mutation. | osimertinib | epidermal growth factor receptor | Homo sapiens |
3 | BACKGROUND: Osimertinib (AZD9291) is an oral, potent, irreversible EGFR tyrosine-kinase inhibitor selective for EGFR tyrosine-kinase inhibitor sensitising mutations, and the EGFR Thr790Met resistance mutation. | osimertinib | epidermal growth factor receptor | Homo sapiens |
4 | BACKGROUND: Osimertinib (AZD9291) is an oral, potent, irreversible EGFR tyrosine-kinase inhibitor selective for EGFR tyrosine-kinase inhibitor sensitising mutations, and the EGFR Thr790Met resistance mutation. | osimertinib | epidermal growth factor receptor | Homo sapiens |
5 | We assessed the efficacy and safety of osimertinib in patients with EGFR Thr790Met-positive non-small-cell lung cancer (NSCLC), who had progressed after previous therapy with an approved EGFR tyrosine-kinase inhibitor. | osimertinib | epidermal growth factor receptor | Homo sapiens |
6 | INTERPRETATION: Osimertinib showed clinical activity with manageable side-effects in patients with EGFR Thr790Met-positive NSCLC. | osimertinib | epidermal growth factor receptor | Homo sapiens |
7 | Therefore, osimertinib could be a suitable treatment for patients with EGFR Thr790Met-positive disease who have progressed on an EGFR tyrosine-kinase inhibitor. | osimertinib | epidermal growth factor receptor | Homo sapiens |
8 | Therefore, osimertinib could be a suitable treatment for patients with EGFR Thr790Met-positive disease who have progressed on an EGFR tyrosine-kinase inhibitor. | osimertinib | epidermal growth factor receptor | Homo sapiens |