Pub. Date : 2016 Nov
PMID : 27594653
3 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
1 | Based on a computational analysis we established HEK293 cell lines overexpressing the mutant OATP1B1 proteins HEK-OATP1B1p.H54Q, -p.H54A, -p.Y169H and -p.Y169A and analyzed protein expression, localization and transport kinetics of the four OATP1B1 substrates bromosulfophthalein, estradiaol-17beta-glucuronide, taurocholate and pravastatin. | Taurocholic Acid | solute carrier organic anion transporter family member 1B1 | Homo sapiens |
2 | Based on a computational analysis we established HEK293 cell lines overexpressing the mutant OATP1B1 proteins HEK-OATP1B1p.H54Q, -p.H54A, -p.Y169H and -p.Y169A and analyzed protein expression, localization and transport kinetics of the four OATP1B1 substrates bromosulfophthalein, estradiaol-17beta-glucuronide, taurocholate and pravastatin. | Taurocholic Acid | solute carrier organic anion transporter family member 1B1 | Homo sapiens |
3 | Based on a computational analysis we established HEK293 cell lines overexpressing the mutant OATP1B1 proteins HEK-OATP1B1p.H54Q, -p.H54A, -p.Y169H and -p.Y169A and analyzed protein expression, localization and transport kinetics of the four OATP1B1 substrates bromosulfophthalein, estradiaol-17beta-glucuronide, taurocholate and pravastatin. | Taurocholic Acid | solute carrier organic anion transporter family member 1B1 | Homo sapiens |