Title : Involvement of CYP 3A5 In the Interaction Between Tacrolimus and Nicardipine: A Case Report.

Pub. Date : 2015

PMID : 25968921






2 Functional Relationships(s)
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Protein Name
Organism
1 Tacrolimus is a calcineurin inhibitor primarily metabolized by CYP3A4 and secondarily by CYP3A5. Tacrolimus cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 Increase of tacrolimus trough concentrations is due to the inhibition of CYP3A4. Tacrolimus cytochrome P450 family 3 subfamily A member 4 Homo sapiens