Title : Desformylflustrabromine (dFBr) and [3H]dFBr-Labeled Binding Sites in a Nicotinic Acetylcholine Receptor.

Pub. Date : 2015 Jul

PMID : 25870334






1 Functional Relationships(s)
Download
Sentence
Compound Name
Protein Name
Organism
1 In the presence of agonist, [(3)H]dFBr also photolabeled amino acids in the nAChR extracellular domain within binding pockets identified previously for the nonselective nAChR PAMs galantamine and physostigmine at the canonical alpha-gamma interface containing the transmitter binding sites and at the noncanonical delta-beta subunit interface. Physostigmine cholinergic receptor nicotinic alpha 4 subunit Homo sapiens