Title : P-glycoprotein inhibition by the agricultural pesticide propiconazole and its hydroxylated metabolites: Implications for pesticide-drug interactions.

Pub. Date : 2015 Jan 5

PMID : 25268938






1 Functional Relationships(s)
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1 In NIH-3T3/MDR1 cells, propiconazole (1 and 10muM) led to decreased cellular resistance (chemosensitization) to paclitaxel, a chemotherapeutic drug and known MDR1 substrate. Paclitaxel ATP-binding cassette, sub-family B (MDR/TAP), member 1B Mus musculus