Pub. Date : 2014 Dec 10
PMID : 25261710
2 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
1 | Dipeptide prodrug approach to evade efflux pumps and CYP3A4 metabolism of lopinavir. | Dipeptides | cytochrome P450 3A12 | Canis lupus familiaris |
2 | In the present study, dipeptide prodrug approach was employed to circumvent efflux pumps (P-gp and MRP2) and CYP3A4 mediated metabolism of LPV. | Dipeptides | cytochrome P450 3A12 | Canis lupus familiaris |