Title : Presynaptic calcium channel inhibition underlies CB₁ cannabinoid receptor-mediated suppression of GABA release.

Pub. Date : 2014 Jun 4

PMID : 24899717






2 Functional Relationships(s)
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1 Altering CB1 function by either increasing endocannabinoid production or removing its tonic activity allowed us to demonstrate that CB1 controls GABA release by inhibiting Ca(2+) entry into presynaptic axon terminals via N-type (Cav2.2) Ca(2+) channels. Endocannabinoids cannabinoid receptor 1 (brain) Mus musculus
2 Altering CB1 function by either increasing endocannabinoid production or removing its tonic activity allowed us to demonstrate that CB1 controls GABA release by inhibiting Ca(2+) entry into presynaptic axon terminals via N-type (Cav2.2) Ca(2+) channels. Endocannabinoids cannabinoid receptor 1 (brain) Mus musculus