Title : Effect of P-glycoprotein on the rat intestinal permeability and metabolism of the BDDCS class 1 drug verapamil.

Pub. Date : 2013 Nov 4

PMID : 24044638






4 Functional Relationships(s)
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1 Effect of P-glycoprotein on the rat intestinal permeability and metabolism of the BDDCS class 1 drug verapamil. Verapamil ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus
2 We investigated the effect of inhibiting P-glycoprotein (P-gp) on the in vitro rat intestinal permeability (Papp) and metabolism of the class 1 drug verapamil. Verapamil ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus
3 We investigated the effect of inhibiting P-glycoprotein (P-gp) on the in vitro rat intestinal permeability (Papp) and metabolism of the class 1 drug verapamil. Verapamil ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus
4 The results suggest that P-gp inhibition has an effect on class 1 drug verapamil and class 2 drug atorvastatin Papp in the rat intestine. Verapamil ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus