Title : Impact of CYP3A5 genotype on tacrolimus versus midazolam clearance in renal transplant recipients: new insights in CYP3A5-mediated drug metabolism.

Pub. Date : 2013 Sep

PMID : 24024898






1 Functional Relationships(s)
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1 BACKGROUND & AIM: In vitro studies have identified both midazolam and tacrolimus as dual CYP3A4 and CYP3A5 substrates. Tacrolimus cytochrome P450 family 3 subfamily A member 4 Homo sapiens