Title : Quantitative prediction of repaglinide-rifampicin complex drug interactions using dynamic and static mechanistic models: delineating differential CYP3A4 induction and OATP1B1 inhibition potential of rifampicin.

Pub. Date : 2013 May

PMID : 23393219






2 Functional Relationships(s)
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1 Quantitative prediction of repaglinide-rifampicin complex drug interactions using dynamic and static mechanistic models: delineating differential CYP3A4 induction and OATP1B1 inhibition potential of rifampicin. repaglinide cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 Repaglinide is mainly metabolized by cytochrome P450 enzymes CYP2C8 and CYP3A4, and it is also a substrate to a hepatic uptake transporter, organic anion transporting polypeptide (OATP)1B1. repaglinide cytochrome P450 family 3 subfamily A member 4 Homo sapiens