Title : Targeting carcinoma-associated fibroblasts within the tumor stroma with a fibroblast activation protein-activated prodrug.

Pub. Date : 2012 Sep 5

PMID : 22911669






2 Functional Relationships(s)
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1 METHODS: The efficacy of FAP-activated peptidyl-TG prodrugs was tested in vitro in cell proliferation assays and effects on intracellular calcium in human cancer cell lines. Calcium fibroblast activation protein alpha Homo sapiens
2 Amino acid-12ADT analogs from FAP-cleaved prodrugs, but not uncleaved prodrugs, produced a rapid rise in intracellular calcium within minutes of exposure. Calcium fibroblast activation protein alpha Homo sapiens