Title : Effect of lersivirine co-administration on pharmacokinetics of methadone in healthy volunteers.

Pub. Date : 2012 Nov 1

PMID : 22682979






3 Functional Relationships(s)
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Protein Name
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1 As methadone is metabolized by CYP3A4 and lersivirine is a weak CYP3A4 inducer, it is possible that lersivirine may decrease methadone concentrations. UK 453,061 cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 As methadone is metabolized by CYP3A4 and lersivirine is a weak CYP3A4 inducer, it is possible that lersivirine may decrease methadone concentrations. UK 453,061 cytochrome P450 family 3 subfamily A member 4 Homo sapiens
3 As methadone is metabolized by CYP3A4 and lersivirine is a weak CYP3A4 inducer, it is possible that lersivirine may decrease methadone concentrations. UK 453,061 cytochrome P450 family 3 subfamily A member 4 Homo sapiens