Title : Preparation of 3-substituted-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidin-4-amines as RET kinase inhibitors.

Pub. Date : 2012 May 24

PMID : 22559926






2 Functional Relationships(s)
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1 Preparation of 3-substituted-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidin-4-amines as RET kinase inhibitors. 3-substituted-1-isopropyl-1h-pyrazolo[3,4-d]pyrimidin-4-amines ret proto-oncogene Homo sapiens
2 A series of 3-substituted-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidin-4-amines have been designed, synthesized, and evaluated as RET protein kinase inhibitors. 3-substituted-1-isopropyl-1h-pyrazolo[3,4-d]pyrimidin-4-amines ret proto-oncogene Homo sapiens