Title : Potent and selective aminopyrimidine-based B-Raf inhibitors with favorable physicochemical and pharmacokinetic properties.

Pub. Date : 2012 Mar 22

PMID : 22335519






1 Functional Relationships(s)
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1 Through structure-based design, we discovered a new class of highly potent aminopyrimidine-based B-Raf inhibitors with improved solubility and pharmacokinetic profiles. 2-aminopyrimidine Braf transforming gene Mus musculus