Title : PXR variants and artemisinin use in Vietnamese subjects: frequency distribution and impact on the interindividual variability of CYP3A induction by artemisinin.

Pub. Date : 2012 Apr

PMID : 22252826






3 Functional Relationships(s)
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1 PXR variants and artemisinin use in Vietnamese subjects: frequency distribution and impact on the interindividual variability of CYP3A induction by artemisinin. artemisinin cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 Here, we report the resequencing and genotyping of PXR variants in 75 Vietnamese individuals previously characterized for CYP3A enzyme activity after artemisinin exposure. artemisinin cytochrome P450 family 3 subfamily A member 4 Homo sapiens
3 A trend of significance was observed between the level of CYP3A4 induction by artemisinin and two PXR variants, the 8118C T (Y328Y) and 10719A G variants. artemisinin cytochrome P450 family 3 subfamily A member 4 Homo sapiens