Title : Synthesis and characterization of high-affinity 4,4-difluoro-4-bora-3a,4a-diaza-s-indacene-labeled fluorescent ligands for human β-adrenoceptors.

Pub. Date : 2011 Oct 13

PMID : 21870877






1 Functional Relationships(s)
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1 Imaging studies with this compound further confirmed that it can be employed to selectively label the human beta2-adrenoceptor in single living cells, with receptor-associated binding prevented by preincubation with the nonfluorescent beta2-selective antagonist 3-(isopropylamino)-1-[(7-methyl-4-indanyl)oxy]butan-2-ol (ICI 118551) ( J. Cardiovasc. 3-(isopropylamino)-1-[(7-methyl-4-indanyl)oxy]butan-2-ol adrenoceptor beta 2 Homo sapiens