Title : Chemical inhibitors of cytochrome P450 isoforms in human liver microsomes: a re-evaluation of P450 isoform selectivity.

Pub. Date : 2011 Mar

PMID : 21336516






1 Functional Relationships(s)
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1 The most selective inhibitors available are furafylline (in co-incubation and pre-incubation conditions) for CYP1A2, 2-phenyl-2-(1-piperidinyl)propane (PPP) for CYP2B6, montelukast for CYP2C8, sulfaphenazole for CYP2C9, (-)-N-3-benzyl-phenobarbital for CYP2C19 and quinidine for CYP2D6. 2-phenyl-2-(1-piperidinyl)propane cytochrome P450 family 2 subfamily C member 8 Homo sapiens