Title : Cocktail-substrate assay system for mechanism-based inhibition of CYP2C9, CYP2D6, and CYP3A using human liver microsomes at an early stage of drug development.

Pub. Date : 2009 Jun

PMID : 19480547






1 Functional Relationships(s)
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1 Using this system, we confirmed that multiple CYP inactivation caused by mechanism-based inhibitors such as isoniazid and amiodarone could be detected simultaneously. Isoniazid cytochrome P450 family 4 subfamily F member 3 Homo sapiens