Title : Discovery and SAR of 2-(1-propylpiperidin-4-yl)-1H-benzimidazole-4-carboxamide: A potent inhibitor of poly(ADP-ribose) polymerase (PARP) for the treatment of cancer.

Pub. Date : 2008 Jul 15

PMID : 18541433






3 Functional Relationships(s)
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1 We have developed a series of cyclic amine-containing benzimidazole carboxamide poly(ADP-ribose)polymerase (PARP) inhibitors, with good PARP-1 enzyme potency, as well as cellular potency. benzimidazole poly (ADP-ribose) polymerase family, member 1 Mus musculus
2 We have developed a series of cyclic amine-containing benzimidazole carboxamide poly(ADP-ribose)polymerase (PARP) inhibitors, with good PARP-1 enzyme potency, as well as cellular potency. benzimidazole poly (ADP-ribose) polymerase family, member 1 Mus musculus
3 We have developed a series of cyclic amine-containing benzimidazole carboxamide poly(ADP-ribose)polymerase (PARP) inhibitors, with good PARP-1 enzyme potency, as well as cellular potency. benzimidazole poly (ADP-ribose) polymerase family, member 1 Mus musculus