Title : Induction of nuclear receptors and drug resistance in the brain microvascular endothelial cells treated with antiepileptic drugs.

Pub. Date : 2008 May

PMID : 18473823






2 Functional Relationships(s)
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1 Carbamazepine, phenobarbital and phenytoin induced the highest levels of P-gp and MPRs expression that was associated with increased activation of PXR and CAR receptors as compared to levetiracetam, tiagabine and topiramate. Phenobarbital ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus
2 We conclude that P-gp and MRPs are differently overexpressed in GPNT and RBE4 by various AEDs and both PXR and CAR are involved in the drug-resistant epilepsy induced by carbamazepine, phenobarbital and phenytoin. Phenobarbital ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus