Title : Modulation of trabectedin (ET-743) hepatobiliary disposition by multidrug resistance-associated proteins (Mrps) may prevent hepatotoxicity.

Pub. Date : 2008 Apr 1

PMID : 18191164






1 Functional Relationships(s)
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1 The protection by DEX against trabectedin-mediated cytotoxicity may be attributed, in part, to enhanced Mrp2 biliary excretion and increased metabolism by CYP3A1/2. Trabectedin ATP binding cassette subfamily C member 2 Rattus norvegicus