Title : N-desalkylquetiapine, a potent norepinephrine reuptake inhibitor and partial 5-HT1A agonist, as a putative mediator of quetiapine's antidepressant activity.

Pub. Date : 2008 Sep

PMID : 18059438






1 Functional Relationships(s)
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1 In the mouse tail suspension test, N-Desalkylquetiapine displayed potent antidepressant-like activity in VMAT2 heterozygous mice at doses as low as 0.1 mg/kg. norquetiapine solute carrier family 18 (vesicular monoamine), member 2 Mus musculus