Title : The influence of macrolide antibiotics on the uptake of organic anions and drugs mediated by OATP1B1 and OATP1B3.

Pub. Date : 2007 May

PMID : 17296622






1 Functional Relationships(s)
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1 The IC50 values for the inhibition of OATP1B3-mediated BSP uptake were 11 microM for telithromycin, 32 microM for clarithromycin, 34 microM for erythromycin, and 37 microM for roxithromycin. Clarithromycin solute carrier organic anion transporter family member 1B3 Homo sapiens