Title : Dipeptide proline diphenyl phosphonates are potent, irreversible inhibitors of seprase (FAPalpha).

Pub. Date : 2006 Jul 28

PMID : 16769036






2 Functional Relationships(s)
Download
Sentence
Compound Name
Protein Name
Organism
1 The most potent inhibitor of DPP-IV and seprase was found to be Gly-ProP(OPh)2, which exhibited overall second-order rate constants of inactivation of 5.24 x 105 M-1 min-1 and 1.06 x 104 M-1 min-1 against DPP-IV and seprase, respectively. gly-prop(oph)2 fibroblast activation protein alpha Homo sapiens
2 The most potent inhibitor of DPP-IV and seprase was found to be Gly-ProP(OPh)2, which exhibited overall second-order rate constants of inactivation of 5.24 x 105 M-1 min-1 and 1.06 x 104 M-1 min-1 against DPP-IV and seprase, respectively. gly-prop(oph)2 fibroblast activation protein alpha Homo sapiens