Title : Pharmacokinetics of ruboxistaurin are significantly altered by rifampicin-mediated CYP3A4 induction.

Pub. Date : 2006 Feb

PMID : 16433874






2 Functional Relationships(s)
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1 Pharmacokinetics of ruboxistaurin are significantly altered by rifampicin-mediated CYP3A4 induction. ruboxistaurin cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 CONCLUSIONS: The effect of rifampicin co-administration on the exposure of ruboxistaurin is consistent with ruboxistaurin being a substrate of CYP3A4. ruboxistaurin cytochrome P450 family 3 subfamily A member 4 Homo sapiens