Title : Major effect of pyrrolic N-benzylation in norbinaltorphimine, the selective kappa-opioid receptor antagonist.

Pub. Date : 2005 Mar 10

PMID : 15743210






2 Functional Relationships(s)
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1 Major effect of pyrrolic N-benzylation in norbinaltorphimine, the selective kappa-opioid receptor antagonist. norbinaltorphimine opioid receptor kappa 1 Homo sapiens
2 Similar modification of the kappa-opioid receptor (KOR) antagonist norBNI (1a) and its 17,17"-diNMe analogue (1d), a low potency mu-opioid receptor (MOR) partial agonist, was found to affect predominantly their MOR activity. norbinaltorphimine opioid receptor kappa 1 Homo sapiens