Title : Ziprasidone metabolism, aldehyde oxidase, and clinical implications.

Pub. Date : 2003 Jun

PMID : 12826984






3 Functional Relationships(s)
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1 Two enzyme systems have been implicated in ziprasidone metabolism: the cytosolic enzyme, aldehyde oxidase, catalyzes the predominant reductive pathway, and cytochrome P4503A4 (CYP3A4) is responsible for two alternative oxidation pathways. ziprasidone cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 Two enzyme systems have been implicated in ziprasidone metabolism: the cytosolic enzyme, aldehyde oxidase, catalyzes the predominant reductive pathway, and cytochrome P4503A4 (CYP3A4) is responsible for two alternative oxidation pathways. ziprasidone cytochrome P450 family 3 subfamily A member 4 Homo sapiens
3 Because CYP3A4 only mediates one third of ziprasidone metabolism, the likelihood of interactions between ziprasidone and CYP3A4 inhibitors/ substrates is low. ziprasidone cytochrome P450 family 3 subfamily A member 4 Homo sapiens