Title : Targeted pharmacological depletion of serum amyloid P component for treatment of human amyloidosis.

Pub. Date : 2002 May 16

PMID : 12015594






1 Functional Relationships(s)
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1 In order to intervene in this process we have developed a drug, R-1-[6-[R-2-carboxy-pyrrolidin-1-yl]-6-oxo-hexanoyl]pyrrolidine-2-carboxylic acid, that is a competitive inhibitor of SAP binding to amyloid fibrils. R-1-(6-(R-2-carboxypyrrolidin-1-yl)-6-oxohexanoyl)pyrrolidine-2-carboxylic acid amyloid P component, serum Homo sapiens