Title : Pharmacokinetics, tissue distribution, metabolism, and excretion of celecoxib in rats.

Pub. Date : 2000 May

PMID : 10772629






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1 The pharmacokinetics, tissue distribution, metabolism, and excretion of celecoxib, 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl] benzenesulfonamide, a cyclooxygenase-2 inhibitor, were investigated in rats. Celecoxib prostaglandin-endoperoxide synthase 2 Rattus norvegicus