Title : Estrogen receptor beta activates the human retinoic acid receptor alpha-1 promoter in response to tamoxifen and other estrogen receptor antagonists, but not in response to estrogen.

Pub. Date : 1999 Mar

PMID : 10076999






2 Functional Relationships(s)
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1 ER antagonists inhibited this estrogen induction through both hERalpha and hERbeta, although raloxifene was more potent through ERalpha than ERbeta, and tamoxifen was more potent via ERbeta than ERalpha. Raloxifene Hydrochloride estrogen receptor 2 Homo sapiens
2 Other ER antagonists including raloxifene, ICI-164,384 and ICI-182,780 also acted as agonists through ERbeta via the hRARalpha-1 promoter. Raloxifene Hydrochloride estrogen receptor 2 Homo sapiens