benzenesulfonamide

carbonic anhydrase 9 ; Homo sapiens







19 Article(s)
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1 34443307 Design, Synthesis, Biological Evaluation, and Computational Studies of Novel Tri-Aryl Imidazole-Benzene Sulfonamide Hybrids as Promising Selective Carbonic Anhydrase IX and XII Inhibitors. 2021 Aug 4 1
2 34769000 Inhibition of Carbonic Anhydrase IX Suppresses Breast Cancer Cell Motility at the Single-Cell Level. 2021 Oct 26 1
3 32028060 Synthesis of some N-aroyl-2-oxindole benzenesulfonamide conjugates with carbonic anhydrase inhibitory activity. 2020 Mar 1
4 30826507 Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer cell lines. 2019 Apr 15 1
5 31276899 Application of hydrazino and hydrazido linkers to connect benzenesulfonamides with hydrophilic/phobic tails for targeting the middle region of human carbonic anhydrases active site: Selective inhibitors of hCA IX. 2019 Oct 1 1
6 29566486 Discovery of Benzenesulfonamide Derivatives as Carbonic Anhydrase Inhibitors with Effective Anticonvulsant Action: Design, Synthesis, and Pharmacological Evaluation. 2018 Apr 12 1
7 30452451 Selective inhibition of carbonic anhydrase IX over carbonic anhydrase XII in breast cancer cells using benzene sulfonamides: Disconnect between activity and growth inhibition. 2018 1
8 28001003 Intrinsic Thermodynamics and Structures of 2,4- and 3,4-Substituted Fluorinated Benzenesulfonamides Binding to Carbonic Anhydrases. 2017 Jan 20 1
9 28065499 Benzenesulfonamide bearing imidazothiadiazole and thiazolotriazole scaffolds as potent tumor associated human carbonic anhydrase IX and XII inhibitors. 2017 Feb 1 1
10 28498332 Design, Synthesis, Molecular Docking Analysis, and Carbonic Anhydrase IX Inhibitory Evaluations of Novel N-Substituted-β-d-Glucosamine Derivatives that Incorporate Benzenesulfonamides. 2017 May 12 1
11 25758852 Functionalization of fluorinated benzenesulfonamides and their inhibitory properties toward carbonic anhydrases. 2015 Apr 1
12 24878197 Synthesis and evaluation of (18)F-labeled tertiary benzenesulfonamides for imaging carbonic anhydrase IX expression in tumours with positron emission tomography. 2014 Jul 15 1
13 23151266 In-silico analysis of chromone containing sulfonamide derivatives as human carbonic anhydrase inhibitors. 2013 Jun 1 1
14 23234246 Synthesis and SAR of novel Re/99mTc-labeled benzenesulfonamide carbonic anhydrase IX inhibitors for molecular imaging of tumor hypoxia. 2013 Jan 24 1
15 23290254 Carbonic anhydrase inhibitors: benzenesulfonamides incorporating cyanoacrylamide moieties are low nanomolar/subnanomolar inhibitors of the tumor-associated isoforms IX and XII. 2013 Mar 15 1
16 23429054 Optimization of heterocyclic substituted benzenesulfonamides as novel carbonic anhydrase IX inhibitors and their structure activity relationship. 2013 Apr 2
17 22548333 A QSAR study on novel series of carbonic anhydrase inhibitors hCA IX--tumor-associated (hypoxia). 2012 Jul 1
18 20598552 Coumarinyl-substituted sulfonamides strongly inhibit several human carbonic anhydrase isoforms: solution and crystallographic investigations. 2010 Jul 15 1
19 15780637 Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II. 2005 Apr 1 1