| 1 |
34814141 | Pregnane-Oximino-Alkyl-Amino-Ether Compound as a Novel Class of TGR5 Receptor Agonist Exhibiting Antidiabetic and Anti-Dyslipidemic Activities. | 2022 |
1 |
| 2 |
33524991 | A Powerful HPLC-ELSD Method for Simultaneous Determination of Fecal Bile Acids in T2DM Rats Interfered by Sanhuang Xiexin Tang. | 2021 Sep 29 |
3 |
| 3 |
33531049 | TGR5 activation attenuates neuroinflammation via Pellino3 inhibition of caspase-8/NLRP3 after middle cerebral artery occlusion in rats. | 2021 Feb 2 |
2 |
| 4 |
31957105 | TGR5 receptor activation attenuates diabetic retinopathy through suppression of RhoA/ROCK signaling. | 2020 Mar |
2 |
| 5 |
32443832 | Hepatic Bile Acid Reuptake in the Rat Depends on Bile Acid Conjugation but Not on Agonistic Properties towards FXR and TGR5. | 2020 May 20 |
4 |
| 6 |
32485177 | Bile Acids Signal via TGR5 to Activate Intestinal Stem Cells and Epithelial Regeneration. | 2020 Sep |
1 |
| 7 |
32699194 | Satiety induced by bile acids is mediated via vagal afferent pathways. | 2020 Jul 23 |
2 |
| 8 |
32859104 | TGR5 Signaling in Hepatic Metabolic Health. | 2020 Aug 26 |
1 |
| 9 |
29999170 | Distribution of bile acid receptor TGR5 in the gastrointestinal tract of dogs. | 2019 Jan |
1 |
| 10 |
31201552 | Obeticholic Acid: An Update of Its Pharmacological Activities in Liver Disorders. | 2019 |
2 |
| 11 |
31493504 | Activation of TGR5 with INT-777 attenuates oxidative stress and neuronal apoptosis via cAMP/PKCε/ALDH2 pathway after subarachnoid hemorrhage in rats. | 2019 Nov 1 |
1 |
| 12 |
28786523 | The bile acid-sequestering resin sevelamer eliminates the acute GLP-1 stimulatory effect of endogenously released bile acids in patients with type 2 diabetes. | 2018 Feb |
1 |
| 13 |
30372884 | Activation of TGR5 promotes osteoblastic cell differentiation and mineralization. | 2018 Dec |
2 |
| 14 |
30671099 | Crosstalk between FXR and TGR5 controls glucagon-like peptide 1 secretion to maintain glycemic homeostasis. | 2018 Dec |
1 |
| 15 |
28091894 | Mechanisms of Action of Surgical Interventions on Weight-Related Diseases: the Potential Role of Bile Acids. | 2017 Mar |
2 |
| 16 |
28580281 | Glucagon-like peptide-2 promotes gallbladder refilling via a TGR5-independent, GLP-2R-dependent pathway. | 2017 Jun |
1 |
| 17 |
28946907 | The relationship between bile acid concentration, glucagon-like-peptide 1, fibroblast growth factor 15 and bile acid receptors in rats during progression of glucose intolerance. | 2017 Sep 25 |
2 |
| 18 |
26757816 | Activation of Transmembrane Bile Acid Receptor TGR5 Modulates Pancreatic Islet α Cells to Promote Glucose Homeostasis. | 2016 Mar 25 |
1 |
| 19 |
26888164 | Effect of chenodeoxycholic acid and the bile acid sequestrant colesevelam on glucagon-like peptide-1 secretion. | 2016 Jun |
1 |
| 20 |
27402811 | Bile acids evoke placental inflammation by activating Gpbar1/NF-κB pathway in intrahepatic cholestasis of pregnancy. | 2016 Dec |
6 |
| 21 |
27808040 | EndoBarrier gastrointestinal liner. Delineation of underlying mechanisms and clinical effects. | 2016 Nov |
1 |
| 22 |
27833095 | Structural assemblies of the di- and oligomeric G-protein coupled receptor TGR5 in live cells: an MFIS-FRET and integrative modelling study. | 2016 Nov 11 |
2 |
| 23 |
25248001 | Bile acid malabsorption in inflammatory bowel disease. | 2015 Feb |
1 |
| 24 |
25540233 | Upregulation of bile acid receptor TGR5 and nNOS in gastric myenteric plexus is responsible for delayed gastric emptying after chronic high-fat feeding in rats. | 2015 May 15 |
2 |
| 25 |
26884847 | Mechanism of bile acid-regulated glucose and lipid metabolism in duodenal-jejunal bypass. | 2015 |
1 |
| 26 |
24986531 | Postprandial gallbladder emptying in patients with type 2 diabetes: potential implications for bile-induced secretion of glucagon-like peptide 1. | 2014 Oct |
2 |
| 27 |
25404917 | Release of GLP-1 and PYY in response to the activation of G protein-coupled bile acid receptor TGR5 is mediated by Epac/PLC-ε pathway and modulated by endogenous H2S. | 2014 |
3 |
| 28 |
22609541 | FXR signaling in the enterohepatic system. | 2013 Apr 10 |
1 |
| 29 |
23275610 | Postprandial gut hormone responses and glucose metabolism in cholecystectomized patients. | 2013 Feb 15 |
1 |
| 30 |
23729782 | Digestive physiology of the pig symposium: intestinal bile acid sensing is linked to key endocrine and metabolic signaling pathways. | 2013 May |
3 |
| 31 |
23849932 | Effect of maternal cholestasis on TGR5 expression in human and rat placenta at term. | 2013 Sep |
1 |
| 32 |
24222092 | The role of gastrointestinal hormones in hepatic lipid metabolism. | 2013 Nov |
1 |
| 33 |
22821947 | Dipeptidyl peptidase IV inhibition potentiates amino acid- and bile acid-induced bicarbonate secretion in rat duodenum. | 2012 Oct |
1 |
| 34 |
23022524 | Activation of transmembrane bile acid receptor TGR5 stimulates insulin secretion in pancreatic β cells. | 2012 Oct 26 |
2 |
| 35 |
20023205 | Bile alcohols function as the ligands of membrane-type bile acid-activated G protein-coupled receptor. | 2010 Jun |
3 |
| 36 |
20297923 | Utility of the carboxylesterase inhibitor bis-para-nitrophenylphosphate (BNPP) in the plasma unbound fraction determination for a hydrolytically unstable amide derivative and agonist of the TGR5 receptor. | 2010 Jun |
2 |
| 37 |
20300620 | Bile acid-induced arrhythmia is mediated by muscarinic M2 receptors in neonatal rat cardiomyocytes. | 2010 Mar 15 |
1 |
| 38 |
20354075 | Gender-dependent effect of Gpbar1 genetic deletion on the metabolic profiles of diet-induced obese mice. | 2010 Jun |
3 |
| 39 |
19346331 | Bile acids as regulatory molecules. | 2009 Aug |
2 |
| 40 |
18468513 | Expression and function of the bile acid receptor TGR5 in Kupffer cells. | 2008 Jul 18 |
4 |
| 41 |
17326144 | The G-protein coupled bile salt receptor TGR5 is expressed in liver sinusoidal endothelial cells. | 2007 Mar |
1 |
| 42 |
15721318 | Bile acids promote glucagon-like peptide-1 secretion through TGR5 in a murine enteroendocrine cell line STC-1. | 2005 Apr 1 |
4 |
| 43 |
12524422 | A G protein-coupled receptor responsive to bile acids. | 2003 Mar 14 |
1 |