benzimidazole

sarcosine dehydrogenase ; Homo sapiens







19 Article(s)
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Title
Pub. Year
#Total Relationships
1 25352112 Comprehensive Review in Current Developments of Benzimidazole-Based Medicinal Chemistry. 2015 Jul 1
2 25599839 Optimisation of in silico derived 2-aminobenzimidazole hits as unprecedented selective kappa opioid receptor agonists. 2015 Feb 15 1
3 26526214 Discovery of potent, selective, and orally bioavailable inhibitors of interleukin-1 receptor-associate kinase-4. 2015 Dec 1 1
4 24461289 Benzimidazole CB2 agonists: design, synthesis and SAR. 2014 Feb 15 1
5 24533813 Benzimidazole derivatives as kinase inhibitors. 2014 1
6 23360431 Inhibitors of human immunodeficiency virus type 1 (HIV-1) attachment. 12. Structure-activity relationships associated with 4-fluoro-6-azaindole derivatives leading to the identification of 1-(4-benzoylpiperazin-1-yl)-2-(4-fluoro-7-[1,2,3]triazol-1-yl-1h-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione (BMS-585248). 2013 Feb 28 1
7 23544603 Novel research strategies of benzimidazole derivatives: a review. 2013 Aug 1
8 23815580 Novel Research Strategies of Benzimidazole Derivatives: A Review. 2013 Jun 26 1
9 22765895 Discovery and optimization of potent and selective imidazopyridine and imidazopyridazine mTOR inhibitors. 2012 Aug 1 1
10 23058106 Benzimidazole inhibitors of the protein kinase CHK2: clarification of the binding mode by flexible side chain docking and protein-ligand crystallography. 2012 Nov 15 2
11 21185722 Azaindoles as potent CRTH2 receptor antagonists. 2011 Jan 15 1
12 20153189 SAR of PXR transactivation in benzimidazole-based IGF-1R kinase inhibitors. 2010 Mar 1 1
13 20185309 Benzimidazole Thumb Pocket I finger-loop inhibitors of HCV NS5B polymerase: improved drug-like properties through C-2 SAR in three sub-series. 2010 Mar 15 2
14 20545947 Design of potent IGF1-R inhibitors related to bis-azaindoles. 2010 Aug 1
15 19716296 GDC-0449-a potent inhibitor of the hedgehog pathway. 2009 Oct 1 1
16 19769332 Inhibitors of human immunodeficiency virus type 1 (HIV-1) attachment. 5. An evolution from indole to azaindoles leading to the discovery of 1-(4-benzoylpiperazin-1-yl)-2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione (BMS-488043), a drug candidate that demonstrates antiviral activity in HIV-1-infected subjects. 2009 Dec 10 1
17 18242988 Discovery of small molecule benzimidazole antagonists of the chemokine receptor CXCR3. 2008 Mar 1 1
18 16442290 Novel non-benzimidazole chk2 kinase inhibitors. 2006 Apr 1 1
19 8401764 Synthesis and cardiotonic evaluation of R-sulfonyl derivatives of azaheterocycles. 1993 Jan-Feb 1