tariquidar

ATP-binding cassette, subfamily B (MDR/TAP), member 1B ; Rattus norvegicus







23 Article(s)
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1 34496661 Comparative vulnerability of PET radioligands to partial inhibition of P-glycoprotein at the blood-brain barrier: A criterion of choice? 2022 Jan 2
2 35588934 Dose-response assessment of cerebral P-glycoprotein inhibition in vivo with [18F]MC225 and PET. 2022 May 20 2
3 34757711 Novel Thienopyrimidine-Based PET Tracers for P2Y12 Receptor Imaging in the Brain. 2021 Dec 1 1
4 32898790 An original radio-biomimetic approach to synthesize radiometabolites for PET imaging. 2020 Nov - Dec 1
5 31322284 Simultaneous quantification of ondansetron and tariquidar in rat and human plasma using a high performance liquid chromatography-ultraviolet method. 2019 Nov 1
6 30130561 Potentiation of antiseizure and neuroprotective efficacy of standard nerve agent treatment by addition of tariquidar. 2018 Sep 1
7 26454782 5-HT2A receptor SPECT imaging with [¹²³I]R91150 under P-gp inhibition with tariquidar: More is better? 2016 Jan 3
8 26621623 Simultaneous Semimechanistic Population Analyses of Levofloxacin in Plasma, Lung, and Prostate To Describe the Influence of Efflux Transporters on Drug Distribution following Intravenous and Intratracheal Administration. 2016 Feb 1
9 27287416 Increasing nerve agent treatment efficacy by P-glycoprotein inhibition. 2016 Nov 25 2
10 23072492 Pharmacokinetic modeling of P-glycoprotein function at the rat and human blood-brain barriers studied with (R)-[11C]verapamil positron emission tomography. 2012 Oct 16 3
11 23143088 Altered GABAA receptor density and unaltered blood-brain barrier transport in a kainate model of epilepsy: an in vivo study using 11C-flumazenil and PET. 2012 Dec 2
12 21600273 Increasing oxime efficacy by blood-brain barrier modulation. 2011 Sep 25 1
13 21677164 A novel positron emission tomography imaging protocol identifies seizure-induced regional overactivity of P-glycoprotein at the blood-brain barrier. 2011 Jun 15 3
14 19796699 Uptake and binding of the serotonin 5-HT1A antagonist [18F]-MPPF in brain of rats: effects of the novel P-glycoprotein inhibitor tariquidar. 2010 Jan 15 6
15 20016890 Dose-response assessment of tariquidar and elacridar and regional quantification of P-glycoprotein inhibition at the rat blood-brain barrier using (R)-[(11)C]verapamil PET. 2010 May 1
16 20633036 Imaging of P-glycoprotein-mediated pharmacoresistance in the hippocampus: proof-of-concept in a chronic rat model of temporal lobe epilepsy. 2010 Sep 1
17 18632828 Tariquidar-induced P-glycoprotein inhibition at the rat blood-brain barrier studied with (R)-11C-verapamil and PET. 2008 Aug 2
18 18760905 Resistance to antiepileptic drugs and expression of P-glycoprotein in two rat models of status epilepticus. 2008 Nov 1
19 17392402 Region-specific overexpression of P-glycoprotein at the blood-brain barrier affects brain uptake of phenytoin in epileptic rats. 2007 Jul 1
20 17437408 Upregulation of brain expression of P-glycoprotein in MRP2-deficient TR(-) rats resembles seizure-induced up-regulation of this drug efflux transporter in normal rats. 2007 Apr 2
21 16650133 Inhibition of the multidrug transporter P-glycoprotein improves seizure control in phenytoin-treated chronic epileptic rats. 2006 Apr 1
22 16928449 The multidrug transporter hypothesis of drug resistance in epilepsy: Proof-of-principle in a rat model of temporal lobe epilepsy. 2006 Oct 1
23 17027274 Determinants of drug brain uptake in a rat model of seizure-associated malformations of cortical development. 2006 Dec 1