ZM 241385

adenosine A2a receptor ; Homo sapiens







27 Article(s)
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Pub. Year
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1 35455444 Beneficial Effects of Polydeoxyribonucleotide (PDRN) in an In Vitro Model of Fuchs Endothelial Corneal Dystrophy. 2022 Apr 3 1
2 34311536 PDRN, a natural bioactive compound, blunts inflammation and positively reprograms healing genes in an "in vitro" model of oral mucositis. 2021 Jun 1
3 33247190 Ligand-directed covalent labelling of a GPCR with a fluorescent tag in live cells. 2020 Nov 27 1
4 30301599 Cervical cancer cells produce TGF-β1 through the CD73-adenosine pathway and maintain CD73 expression through the autocrine activity of TGF-β1. 2019 Jun 1
5 30657045 Adenosine Analogues as Opposite Modulators of the Cisplatin Resistance of Ovarian Cancer Cells. 2019 1
6 30907983 Adenosine from a biologic source regulates neutrophil extracellular traps (NETs). 2019 Jun 1
7 28167788 Crystal structure of the adenosine A2A receptor bound to an antagonist reveals a potential allosteric pocket. 2017 Feb 21 2
8 26631535 Stimulation of adenosine A2A receptors reduces intracellular cholesterol accumulation and rescues mitochondrial abnormalities in human neural cell models of Niemann-Pick C1. 2016 Apr 1
9 26873858 Molecular Basis of Ligand Dissociation from the Adenosine A2A Receptor. 2016 May 1
10 27096000 Inhibition of Gαs/cAMP Signaling Decreases TCR-Stimulated IL-2 transcription in CD4(+) T Helper Cells. 2015 Jul 6 2
11 24591302 Binding kinetics of ZM241385 derivatives at the human adenosine A2A receptor. 2014 Apr 2
12 25179165 Diadenosine diphosphate (Ap₂A) delays neutrophil apoptosis via the adenosine A2A receptor and cAMP/PKA pathway. 2014 Oct 1
13 23332700 Crystallogenesis of adenosine A(2A) receptor-T4 lysozyme fusion protein: a practical route for the structure. 2013 1
14 23593569 SKCa Channels Blockage Increases the Expression of Adenosine A2A Receptor in Jurkat Human T Cells. 2013 Apr 1
15 23637137 Adenosine A(2A) receptors regulate the activity of sleep regulatory GABAergic neurons in the preoptic hypothalamus. 2013 Jul 1 1
16 23933651 Modulation of A₂a receptor antagonist on D₂ receptor internalization and ERK phosphorylation. 2013 Oct 2
17 20595055 Structural features of adenosine receptors: from crystal to function. 2011 May 1
18 21501622 Thermostabilisation of an agonist-bound conformation of the human adenosine A(2A) receptor. 2011 Jun 10 1
19 21970461 Computational study of the binding modes of caffeine to the adenosine A2A receptor. 2011 Dec 1 1
20 20063437 GPCR 3D homology models for ligand screening: lessons learned from blind predictions of adenosine A2a receptor complex. 2010 Jan 2
21 18603240 Adenosine A(2A) receptor dynamics studied with the novel fluorescent agonist Alexa488-APEC. 2008 Aug 20 1
22 19035488 Atheroprotective effects of methotrexate on reverse cholesterol transport proteins and foam cell transformation in human THP-1 monocyte/macrophages. 2008 Dec 1
23 17474152 Adenosine closes the K+ channel KCa3.1 in human lung mast cells and inhibits their migration via the adenosine A2A receptor. 2007 Jun 1
24 17575165 Inhibition of cytokine production and cytotoxic activity of human antimelanoma specific CD8+ and CD4+ T lymphocytes by adenosine-protein kinase A type I signaling. 2007 Jun 15 1
25 17705048 Adenosine inhibition of lipopolysaccharide-induced interleukin-6 secretion by the osteoblastic cell line MG-63. 2007 Oct 1
26 16274777 Adenosine prevents neutrophil adhesion to human endothelial cells after hypoxia/reoxygenation. 2005 Dec 7 1
27 12970092 Brief, repeated, oxygen-glucose deprivation episodes protect neurotransmission from a longer ischemic episode in the in vitro hippocampus: role of adenosine receptors. 2003 Sep 1