darolutamide

androgen receptor ; Homo sapiens







42 Article(s)
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1 34449248 A New Old Target: Androgen Receptor Signaling and Advanced Prostate Cancer. 2022 Jan 6 3
2 34866168 Clinical Pharmacokinetics of the Androgen Receptor Inhibitor Darolutamide in Healthy Subjects and Patients with Hepatic or Renal Impairment. 2022 Apr 3
3 35179323 Darolutamide and Survival in Metastatic, Hormone-Sensitive Prostate Cancer. 2022 Mar 24 1
4 35184345 A case of skin rash during oral administration of a novel androgen receptor inhibitor, darolutamide. 2022 Jul 1
5 35201849 A Case of Prostate Cancer Harboring Androgen Receptor T878A Progesterone-Responsive Mutant Emerging After Abiraterone Acetate Treatment Responding to Darolutamide. 2022 Feb 1
6 35343943 Cases in the management of nonmetastatic castration-resistant prostate cancer: darolutamide as the first androgen receptor inhibitor in a fit, older man. 2022 Jan 1
7 35390118 Targeting the androgen receptor signaling pathway in advanced prostate cancer. 2022 Apr 7 2
8 35490582 Development of novel androgen receptor antagonists based on the structure of darolutamide. 2022 Jul 3
9 35553247 Decisions and dilemmas in non-metastatic castration-resistant prostate cancer management. 2022 May 13 1
10 35579577 Factors that guide selection among androgen receptor inhibitors in patients with nonmetastatic castration-resistant prostate cancer. 2022 May 1
11 32881669 Darolutamide as a Second-Generation Androgen Receptor Inhibitor in the Treatment of Prostate Cancer. 2021 9
12 32958445 Androgen receptor inhibitor treatments: Cardiovascular adverse events and comorbidity considerations in patients with non-metastatic prostate cancer. 2021 Jan 1
13 33135506 An up-to-date evaluation of darolutamide for the treatment of prostate cancer. 2021 Mar 1
14 33140306 Endocrine consequences of treatment with the new androgen receptor axis-targeted agents for advanced prostate cancer. 2021 Mar 1
15 33785516 Metabolism and Mass Balance of the Novel Nonsteroidal Androgen Receptor Inhibitor Darolutamide in Humans. 2021 Jun 1
16 34128827 Androgen receptor signaling inhibitors: post-chemotherapy, pre-chemotherapy and now in castration-sensitive prostate cancer. 2021 Jul 15 1
17 34208290 Evaluation of Darolutamide (ODM201) Efficiency on Androgen Receptor Mutants Reported to Date in Prostate Cancer Patients. 2021 Jun 11 2
18 34362254 Current treatment of non-metastatic castration-refractory prostate cancer. 2021 Spring 1
19 34526701 Neoadjuvant hormonal therapy before radical prostatectomy in high-risk prostate cancer. 2021 Dec 1
20 34884545 Delineating the Molecular Events Underlying Development of Prostate Cancer Variants with Neuroendocrine/Small Cell Carcinoma Characteristics. 2021 Nov 25 1
21 31844181 A review of prostate cancer treatment impact on the CNS and cognitive function. 2020 Jun 1
22 32333502 Darolutamide antagonizes androgen signaling by blocking enhancer and super-enhancer activation. 2020 Sep 7
23 32456317 Second-Generation Androgen Receptor Antagonists as Hormonal Therapeutics for Three Forms of Prostate Cancer. 2020 May 24 1
24 32549073 Clinical and Surgical Assistance in Prostate Cancer during the COVID-19 Pandemic: Implementation of assistance protocols. 2020 Jul 1
25 32562083 Interleukin-23 Represses the Level of Cell Senescence Induced by the Androgen Receptor Antagonists Enzalutamide and Darolutamide in Castration-Resistant Prostate Cancer Cells. 2020 Aug 1
26 32765070 Darolutamide: An Evidenced-Based Review of Its Efficacy and Safety in the Treatment of Prostate Cancer. 2020 2
27 32823970 Deep Learning Modeling of Androgen Receptor Responses to Prostate Cancer Therapies. 2020 Aug 14 2
28 33237495 Darolutamide: A Review in Non-Metastatic Castration-Resistant Prostate Cancer. 2020 Dec 4
29 30115959 Non-metastatic castration resistant prostate cancer: a review of current and emerging medical therapies. 2019 Mar 1
30 30824428 Darolutamide Slows Metastasis in Prostate Cancer. 2019 Apr 1
31 30828788 Darolutamide is a potent androgen receptor antagonist with strong efficacy in prostate cancer models. 2019 Sep 1 8
32 31437779 Discovery and biological evaluation of darolutamide derivatives as inhibitors and down-regulators of wild-type AR and the mutants. 2019 Nov 15 2
33 31471641 [A new androgen receptor antagonist : Darolutamide for patients with non-metastatic castration-resistant prostate cancer]. 2019 Oct 1
34 31571146 Drug-Drug Interaction Potential of Darolutamide: In Vitro and Clinical Studies. 2019 Dec 2
35 31605368 Darolutamide: First Approval. 2019 Nov 2
36 32073798 [Androgen receptor inhibitors in prostate cancer: new drugs, but for which patient?] 2019 Nov 28 1
37 28851578 Moving Towards Precision Urologic Oncology: Targeting Enzalutamide-resistant Prostate Cancer and Mutated Forms of the Androgen Receptor Using the Novel Inhibitor Darolutamide (ODM-201). 2018 Jan 10
38 30197098 Clinical Development of Darolutamide: A Novel Androgen Receptor Antagonist for the Treatment of Prostate Cancer. 2018 Oct 2
39 28490267 Darolutamide (ODM-201) for the treatment of prostate cancer. 2017 Jun 2
40 26137992 Discovery of ODM-201, a new-generation androgen receptor inhibitor targeting resistance mechanisms to androgen signaling-directed prostate cancer therapies. 2015 Jul 3 5
41 26313416 ODM-201: a new-generation androgen receptor inhibitor in castration-resistant prostate cancer. 2015 1
42 24974051 Activity and safety of ODM-201 in patients with progressive metastatic castration-resistant prostate cancer (ARADES): an open-label phase 1 dose-escalation and randomised phase 2 dose expansion trial. 2014 Aug 4