Title : PBPK Modeling of Coproporphyrin I as an Endogenous Biomarker for Drug Interactions Involving Inhibition of Hepatic OATP1B1 and OATP1B3.

Pub. Date : 2018 Nov

PMID : 30175555






1 Functional Relationships(s)
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1 The in vivo inhibition constants of rifampicin used as initial input parameters for OATP1Bs (Ki,u,OATP1Bs ) and multidrug resistance-associated protein two-mediated biliary excretion were estimated as 0.23 and 0.87 muM, respectively, from previous reports. Rifampin ornithine aminotransferase pseudogene 1 Homo sapiens