Title : Iptakalim, a vascular ATP-sensitive potassium (KATP) channel opener, closes rat pancreatic beta-cell KATP channels and increases insulin release.

Pub. Date : 2007 Aug

PMID : 17522344






1 Functional Relationships(s)
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1 Finally, iptakalim inhibited Kir6.2/SUR1, but it activated Kir6.1/SUR2B (vascular-type), K(ATP) channels heterologously expressed in Xenopus oocytes. N-(1-methylethyl)-1,1,2-trimethylpropylamine potassium inwardly rectifying channel subfamily J member 8 L homeolog Xenopus laevis