Title : Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. Part 2: Optimization of 5,8-disubstituted derivatives.

Pub. Date : 2004 Sep 20

PMID : 15324877






2 Functional Relationships(s)
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1 Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. spiroquinazolinones phosphodiesterase 7A Homo sapiens
2 The optimization of 5,8-disubstituted spirocyclohexane-quinazolinones into potent, selective, soluble PDE7 inhibitors with acceptable in vivo pharmacokinetic parameters is presented. 5,8-disubstituted spirocyclohexane-quinazolinones phosphodiesterase 7A Homo sapiens