Title : Lack of pharmacokinetic or pharmacodynamic interaction between memantine and donepezil.

Pub. Date : 2004 Sep

PMID : 15266045






3 Functional Relationships(s)
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1 OBJECTIVE: To determine whether an in vivo pharmacokinetic interaction exists between memantine and the acetylcholinesterase (AChE) inhibitor donepezil. Memantine acetylcholinesterase (Cartwright blood group) Homo sapiens
2 OBJECTIVE: To determine whether an in vivo pharmacokinetic interaction exists between memantine and the acetylcholinesterase (AChE) inhibitor donepezil. Memantine acetylcholinesterase (Cartwright blood group) Homo sapiens
3 In addition, AChE inhibition was measured in red blood cells by radiolabeled-enzyme assay following administration of donepezil alone and after a single memantine dose. Memantine acetylcholinesterase (Cartwright blood group) Homo sapiens