Title : Peptoid CCK receptor antagonists: pharmacological evaluation of CCKA, CCKB and mixed CCKA/B receptor antagonists.

Pub. Date : 1995 Nov 14

PMID : 8605955






1 Functional Relationships(s)
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1 The pyrazolidinone PD 141479 (trans-5-(2-chlorophenyl)-3-oxo-4-phenyl-N-[4- (trifluoromethyl)phenyl]-1-pyrazolidinecarboxamide) was found to interact selectively with the CCKB receptor (CCKB IC50 = 36 nM, CCKA IC50 = 1100 nM). trans-5-(2-chlorophenyl)-3-oxo-4-phenyl-n-[4- (trifluoromethyl)phenyl]-1-pyrazolidinecarboxamide cholecystokinin B receptor Rattus norvegicus