Title : S-methyl N,N-diethylthiocarbamate sulfone, a potential metabolite of disulfiram and potent inhibitor of low Km mitochondrial aldehyde dehydrogenase.

Pub. Date : 1995 Mar 1

PMID : 7887984






1 Functional Relationships(s)
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1 The substrate (acetaldehyde, 80 microM) and cofactor (NAD, 0.5 mM) together completely protected ALDH from inhibition by MeDTC sulfone; substrate alone partially protected the enzyme. NAD aldehyde dehydrogenase 3 family, member A1 Rattus norvegicus