Title : Design and synthesis of marine sesterterpene analogues as novel estrogen receptor α degraders for breast cancer treatment.

Pub. Date : 2022 Feb 5

PMID : 34992039






2 Functional Relationships(s)
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1 Design and synthesis of marine sesterterpene analogues as novel estrogen receptor alpha degraders for breast cancer treatment. Sesterterpenes estrogen receptor 1 Homo sapiens
2 The marine sesterterpene compound MHO7 had been reported to be a potential ERalpha degradation agent. Sesterterpenes estrogen receptor 1 Homo sapiens