Title : Accelerating Clinical Development of Idasanutlin through a Physiologically Based Pharmacokinetic Modeling Risk Assessment for CYP450 Isoenzyme-Related Drug-Drug Interactions.

Pub. Date : 2022 Mar

PMID : 34937801






1 Functional Relationships(s)
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1 Idasanutlin"s clearance is dependent on CYP3A4/2C8, forming its major circulating metabolite M4, with contributions from UGT1A3 and biliary excretion. RG7388 UDP glucuronosyltransferase family 1 member A3 Homo sapiens